Short and Efficient Synthesis of Optically Active N-Tosyl.
Aziridines (azacyclopropanes) constitute the well-known class of heterocyclic compounds. The studies on synthesis and reactivity of aziridines have drawn tremendous interest of organic chemists. The main feature of interest in the chemistry of this molecule is the ring-strain associated with it.Aziridines are attractive and versatile building blocks in organic synthesis and medicinal chemistry because they allow convenient access to useful nitrogen-containing biologically active compounds.SYNTHESIS OF IMIDAZOLINES FROM AZIRIDINES By Michael Robert Kuszpit The majority of the work in this thesis presents a new method to syntheisize imidazolines from both chiral and racemic aziridines. The purpose of synthesizing such heterocycles was for there known biological activity. Previous research in the Tepe group has.
A novel and efficient domino procedure has been developed for the synthesis of 1,4-benzothiazepin-5-ones from simple and readily accessible N-tosyl aziridines and o-iodothiophenols. This process involves aziridines ring-opening with o-iodothiophenols, followed by palladium-catalyzed intramolecular carboxamidation.Tosyl aziridine synthesis essay 911 essay papers on trust sue bentley author biography essay writing as punishment research paper unitarisme dan federalisme dissertation entertainment during the great depression essay writing an essay based on a picture gm essay shazia ilmi swachh bharat essay.
Aziridines, Building Blocks, Chemical Synthesis, Nitrogen Compounds - Organic Building Blocks, Organic Building Blocks.
